The Biological Testing Branch conducted a literature search in August 2008 to determine the number of
references that existed for mouse xenografts associated with these agents. The search was conducted
using the SciFinder® 2007 database search tool with the following criteria selected: [1] includes
journals, reviews, conferences, and clinical trials; [2] excludes patents; [3] the keywords were compound
name, xenograft, mouse; and [4] includes word combinations that were present and/or all concepts to be
found in cited references.
| AGENT |
YEAR INTRODUCED |
# OF REFERENCES YIELDED |
| PDF |
Text Only |
|
|
| PPI-2458 [abarelix, plenaxis] |
PPI-2458 [abarelix, plenaxis] |
2004 |
1 |
| aclarubicin |
aclarubicin |
1981 |
4 |
| actinomycin D |
actinomycin D |
1964 |
10 |
| aldesleukin |
aldesleukin |
1992 |
1 |
| alemtuzumab |
alemtuzumab |
2001 |
1 |
| alitretinoin |
alitretinoin |
1999 |
10 |
| aminoglutethimide |
aminoglutethimide |
1981 |
5 |
| amrubicin HCl |
amrubicin HCl |
2002 |
5 |
| amsacrine |
amsacrine |
1987 |
21 |
| anastrozole |
anastrozole |
1995 |
2 |
| angiotensin II |
angiotensin II |
1994 |
8 |
| arglabin |
|
1999 |
0 |
| arsenic trioxide |
arsenic trioxide |
2000 |
12 |
| asparaginase |
asparaginase |
1969 |
6 |
| azacytidine |
azacytidine |
Pre-1977 |
2 |
| bcg live |
|
1990 |
0 |
| CKD-602 [belotecan hydrocholoride] |
CKD-602 [belotecan hydrocholoride] |
2004 |
2 |
| bevacizumab |
bevacizumab |
2004 |
15 |
| bexarotene |
bexarotene |
2000 |
11 |
| bicalutamide |
bicalutamide |
1995 |
3 |
| bisantrene hydrochloride |
bisantrene hydrochloride |
1990 |
1 |
| bleomycin |
bleomycin |
1966 |
26 |
| bortezomib |
bortezomib |
2003 |
14 |
| busulfan |
busulfan |
1954 |
7 |
| calusterone [dimethyltestosterone] |
|
1973 |
0 |
| camostat mesylate |
camostat mesylate |
1985 |
1 |
| capecitabine |
capecitabine |
1998 |
20 |
| carboplatin |
carboplatin |
1986 |
40 |
| carmofur |
carmofur |
1981 |
11 |
| carmustine [BCNU] |
carmustine [BCNU] |
1977 |
48 |
| carzinophilin [carzinophyllin] |
|
1954 |
0 |
| celmoleukin [tucotuzumab, EMD273066] |
|
1992 |
0 |
| cetuximab |
cetuximab |
2003 |
27 |
| chlorambucil |
chlorambucil |
1956 |
2 |
| TACE [chlortrianisene, trioxifene, LY133314] |
TACE [chlortrianisene, trioxifene, LY133314] |
Pre-1981 |
1 |
| chromomycin A3 |
chromomycin A3 |
1961 |
4 |
| cis-diamminedichloroplatinum |
cis-diamminedichloroplatinum |
1979 |
116 |
| cladribine |
cladribine |
1993 |
4 |
| clofarabine |
clofarabine |
2005 |
2 |
| cyclophosphamide |
cyclophosphamide |
1957 |
101 |
| cytarabine ocfosfate |
cytarabine ocfosfate |
1993 |
1 |
| cytosine arabinoside |
cytosine arabinoside |
1969 |
16 |
| DTIC [dacarbazine] |
DTIC [dacarbazine] |
1975 |
11 |
| dasatinib |
dasatinib |
2006 |
3 |
| daunomycin |
daunomycin |
1967 |
7 |
| decitabine |
decitabine |
2006 |
12 |
| ONTAK [denileukin diftitox, DAB389 IL-2] |
ONTAK [denileukin diftitox, DAB389 IL-2] |
1999 |
1 |
| dexamethasone |
dexamethasone |
1958 |
15 |
| diethylstilbestrol |
diethylstilbestrol |
Pre-1970 |
15 |
| docetaxel |
docetaxel |
1995 |
68 |
| doxifluridine |
doxifluridine |
1987 |
54 |
| doxorubicin |
doxorubicin |
1966 |
180 |
| dromostanolone [masteron] |
|
1961 |
0 |
| elliptinium acetate |
elliptinium acetate |
1983 |
1 |
| enocitabine |
enocitabine |
1983 |
1 |
| epirubicin HCL |
>epirubicin HCL |
1984 |
6 |
| erlotinib hydrochloride |
erlotinib hydrochloride |
2004 |
14 |
| estramustine |
estramustine |
1980 |
4 |
| ethinyl estradiol [estradiol] |
ethinyl estradiol [estradiol] |
Pre-1970 |
2 [56] |
| etoposide |
etoposide |
1980 |
42 |
| exemestane |
exemestane |
1999 |
5 |
| fadrozole HCL |
fadrozole HCL |
1995 |
1 |
| floxuridine |
floxuridine |
1971 |
66 |
| fludarabine phosphate |
fludarabine phosphate |
1991 |
18 |
| fluorouracil |
fluorouracil |
1962 |
162 |
| fluoxymesterone [halotestin] |
|
Pre-1970 |
0 |
| flutamide |
flutamide |
1983 |
18 |
| formestane |
formestane |
1993 |
6 |
| fosfestrol |
|
Pre-1977 |
0 |
| fotemustine |
fotemustine |
1989 |
6 |
| ftorafur |
ftorafur |
1972 |
92 |
| fulvestrant |
fulvestrant |
2002 |
6 |
| gefitinib |
gefitinib |
2002 |
37 |
| gemcitabine HCL |
gemcitabine HCL |
1995 |
77 |
| gemtuzumab ozogamicin |
gemtuzumab ozogamicin |
2000 |
2 |
| goserelin acetate |
goserelin acetate |
1987 |
1 |
| H-101 [gendicine] |
|
2005 |
0 |
| heptaplatin |
heptaplatin |
1999 |
1 |
| hexamethylmelamine |
hexamethylmelamine |
1979 |
6 |
| hexyl [5] aminolevulinate |
hexyl [5] aminolevulinate |
2004 |
4 |
| histrelin [vantas, supprelin LA] |
|
2004 |
0 |
| hydroxyprogesterone |
hydroxyprogesterone |
Pre-1970 |
3 |
| hydroxyurea |
hydroxyurea |
1968 |
21 |
| idarubicin hydrochloride |
idarubicin hydrochloride |
1990 |
1 |
| ifosfamide |
ifosfamide |
1976 |
15 |
| imatinib |
imatinib |
2001 |
16 |
| interferon alpha-2a |
interferon alpha-2a |
1986 |
7 |
| interferon alpha-2b |
interferon alpha-2b |
1986 |
4 |
| interferon gamma-1a |
interferon gamma-1a |
1992 |
1 |
| interleukin-2 |
interleukin-2 |
1989 |
50 |
| irinotecan |
irinotecan |
1994 |
45 |
| lenalidomide |
lenalidomide |
2005 |
6 |
| letrozole |
letrozole |
1996 |
4 |
| leucovorin |
leucovorin |
1950 |
9 |
| leuprolide |
leuprolide |
1984 |
2 |
| levamisole |
levamisole |
Pre-1981 |
2 |
| lobaplatin |
lobaplatin |
1998 |
1 |
| lomustine [CCNU] |
lomustine [CCNU] |
1976 |
3 [5] |
| lonidamine |
lonidamine |
1987 |
1 |
| nordihydroguaiaretic acid [NDGA, masoprocol, actinex] |
nordihydroguaiaretic acid [NDGA, masoprocol, actinex] |
1992 |
14 |
| nitrogen mustard [mechlorethanamine] |
nitrogen mustard [mechlorethanamine] |
1958 |
46 |
| medroxyprogesterone |
medroxyprogesterone |
1958 |
20 |
| megesterol acetate |
megesterol acetate |
1971 |
1 |
| melanoma theraccine [melacine] |
|
2001 |
0 |
| melphalan |
melphalan |
1961 |
38 |
| mercaptopurine |
mercaptopurine |
1953 |
8 |
| methotrexate |
methotrexate |
1954 |
45 |
| methylprednisolone |
methylprednisolone |
1955 |
10 |
| methyltestosterone |
|
1974 |
0 |
| miltefosine |
miltefosine |
1993 |
2 |
| mithramycin |
mithramycin |
1961 |
7 |
| mitobronitol |
|
1979 |
0 |
| mitomycin C |
mitomycin C |
1956 |
81 |
| mitotane |
mitotane |
1970 |
1 |
| mitoxantrone |
mitoxantrone |
1984 |
8 |
| mobenakin |
|
1999 |
0 |
| nadrolone phenylpropionate [durabol] |
|
1959 |
0 |
| nafoxidine |
nafoxidine |
Pre-1977 |
1 |
| nedaplatin |
nedaplatin |
1995 |
17 |
| nelarabine [arranon] |
|
2005 |
0 |
| neocarzinostatin |
neocarzinostatin |
1976 |
6 |
| nilutamide |
|
1987 |
0 |
| nimustine |
nimustine |
Pre-1981 |
3 |
| norethindrone |
norethindrone |
Pre-1977 |
1 |
| oxaliplatin |
oxaliplatin |
1996 |
16 |
| paclitaxel |
paclitaxel |
1993 |
162 |
| paclitaxel nanoparticles |
paclitaxel nanoparticles |
2005 |
2 |
| pamidronate |
pamidronate |
1987 |
4 |
| pegaspargase |
|
1994 |
0 |
| pemetrexed |
pemetrexed |
2004 |
2 |
| pentostatin [deoxycoformycin, nipent] |
|
1992 |
0 |
| peplomycin |
peplomycin |
1981 |
16 |
| pipobroman [vercyte, NSC 25154] |
|
1966 |
0 |
| pirarubicin |
pirarubicin |
1988 |
15 |
| porfimer sodium |
porfimer sodium |
1993 |
7 |
| prednisolone |
prednisolone |
Pre-1977 |
2 |
| prednisone |
prednisone |
Pre-1970 |
12 |
| procarbazine |
procarbazine |
1969 |
6 |
| raltitrexed |
raltitrexed |
1996 |
14 |
| ranimustine |
ranimustine |
1987 |
1 |
| razoxane |
razoxane |
Pre-1977 |
6 |
| rituximab |
rituximab |
1997 |
19 |
| sarkomycin |
|
1954 |
0 |
| semustine |
semustine |
Pre-1977 |
27 |
| sobuzoxane |
sobuzoxane |
1994 |
3 |
| solamargine [coramsine] |
|
1987 |
0 |
| sorafenib |
sorafenib |
2005 |
5 |
| streptozocin |
streptozocin |
Pre-1977 |
3 |
| sunitinib |
sunitinib |
2006 |
4 |
| tamibarotene |
tamibarotene |
2005 |
1 |
| tamoxifen |
tamoxifen |
1973 |
64 |
| Tumor necrosis factor alpha/a [tasonermin, beromun] |
Tumor necrosis factor alpha/a [tasonermin, beromun] |
1999 |
10 |
| teceleukin [human IL-2 immunace] |
|
1992 |
0 |
| temozolomide |
temozolomide |
1999 |
30 |
| teniposide |
teniposide |
1967 |
2 |
| testolactone [teslac, fludestrin] |
|
1969 |
0 |
| testosterone |
testosterone |
Pre-1970 |
24 |
| thioguanine |
thioguanine |
1966 |
8 |
| thiotepa |
thiotepa |
1959 |
4 |
| topotecan |
topotecan |
1996 |
46 |
| toremifene |
toremifene |
1989 |
1 |
| tositumomab |
tositumomab |
2003 |
3 |
| trastuzumab |
trastuzumab |
1998 |
36 |
| triamcinolone |
triamcinolone |
1958 |
5 |
| triethylenemelamine [TEM] |
|
Pre-1981 |
0 |
| triptorelin |
triptorelin |
1986 |
4 |
| uracil mustard [uramustine] |
|
1966 |
0 |
| valrubicin |
valrubicin |
1999 |
4 |
| vapreotide |
vapreotide |
2003 |
20 |
| vinblastine |
vinblastine |
1965 |
30 |
| vincristine |
vincristine |
1963 |
49 |
| vindesine |
vindesine |
1979 |
14 |
| vinorelbine |
vinorelbine |
1989 |
17 |
| zinostatin stimalamer [YM881, SMANCS] |
|
1994 |
0 |
| zoledronic acid |
zoledronic acid |
2000 |
19 |