Anti-cancer Agents by Mechanism
Alkylating Agents
| Asaley | NSC 167780 |
| AZQ | NSC 182986 |
| BCNU | NSC 409962 |
| Busulfan | NSC 750 |
| carboxyphthalatoplatinum | NSC 271674 |
| CBDCA | NSC 241240 |
| CCNU | NSC 79037 |
| CHIP | NSC 256927 |
| chlorambucil | NSC 3088 |
| chlorozotocin | NSC 178248 |
| cis-platinum | NSC 119875 |
| clomesone | NSC 338947 |
| cyanomorpholinodoxorubicin | NSC 357704 |
| cyclodisone | NSC 348948 |
| dianhydrogalactitol | NSC 132313 |
| fluorodopan | NSC 73754 |
| hepsulfam | NSC 329680 |
| hycanthone | NSC 142982 |
| melphalan | NSC 8806 |
| methyl CCNU | NSC 95441 |
| mitomycin C | NSC 26980 |
| mitozolamide | NSC 353451 |
| nitrogen mustard | NSC 762 |
| PCNU | NSC 95466 |
| piperazine ../drugs/mainator | NSC 344007 |
| piperazinedione | NSC 135758 |
| pipobroman | NSC 25154 |
| porfiromycin | NSC 56410 |
| spirohydantoin mustard | NSC 172112 |
| teroxirone | NSC 296934 |
| tetraplatin | NSC 363812 |
| thio-tepa | NSC 6396 |
| triethylenemelamine | NSC 9706 |
| uracil nitrogen mustard | NSC 34462 |
| Yoshi-864 | NSC 102627 |
Antimitotic Agents
| allocolchicine | NSC 406042 |
| Halichondrin B | NSC 609395 |
| colchicine | NSC 757 |
| colchicine derivative | NSC 33410 |
| dolastatin 10 | NSC 376128 |
| maytansine | NSC 153858 |
| rhizoxin | NSC 332598 |
| taxol | NSC 125973 |
| taxol derivative | NSC 608832 |
| thiocolchicine | NSC 361792 |
| trityl cysteine | NSC 83265 |
| vinblastine sulfate | NSC 49842 |
| vincristine sulfate | NSC 67574 |
Topoisomerase I Inhibitors
| camptothecin | NSC 94600 |
| camptothecin, Na salt | NSC 100880 |
| aminocamptothecin | NSC 603071 |
| camptothecin derivative | NSC 95382 |
| camptothecin derivative | NSC 107124 |
| camptothecin derivative | NSC 643833 |
| camptothecin derivative | NSC 629971 |
| camptothecin derivative | NSC 295500 |
| camptothecin derivative | NSC 249910 |
| camptothecin derivative | NSC 606985 |
| camptothecin derivative | NSC 374028 |
| camptothecin derivative | NSC 176323 |
| camptothecin derivative | NSC 295501 |
| camptothecin derivative | NSC 606172 |
| camptothecin derivative | NSC 606173 |
| camptothecin derivative | NSC 610458 |
| camptothecin derivative | NSC 618939 |
| camptothecin derivative | NSC 610457 |
| camptothecin derivative | NSC 610459 |
| camptothecin derivative | NSC 606499 |
| camptothecin derivative | NSC 610456 |
| camptothecin derivative | NSC 364830 |
| camptothecin derivative | NSC 606497 |
| morpholinodoxorubicin | NSC 354646 |
Topoisomerase II Inhibitors
| doxorubicin | NSC 123127 |
| amonafide | NSC 308847 |
| m-AMSA | NSC 249992 |
| anthrapyrazole derivative | NSC 355644 |
| pyrazoloacridine | NSC 366140 |
| bisantrene HCL | NSC 337766 |
| daunorubicin | NSC 82151 |
| deoxydoxorubicin | NSC 267469 |
| mitoxantrone | NSC 301739 |
| menogaril | NSC 269148 |
| N,N-dibenzyl daunomycin | NSC 268242 |
| oxanthrazole | NSC 349174 |
| rubidazone | NSC 164011 |
| VM-26 | NSC 122819 |
| VP-16 | NSC 141540 |
RNA/DNA Antimetabolites
| L-alanosine | NSC 153353 |
| 5-azacytidine | NSC 102816 |
| 5-fluorouracil | NSC 19893 |
| acivicin | NSC 163501 |
| aminopterin derivative | NSC 132483 |
| aminopterin derivative | NSC 184692 |
| aminopterin derivative | NSC 134033 |
| an antifol | NSC 623017 |
| Baker's soluble antifol | NSC 139105 |
| dichlorallyl lawsone | NSC 126771 |
| brequinar | NSC 368390 |
| ftorafur (pro-drug) | NSC 148958 |
| 5,6-dihydro-5-azacytidine | NSC 264880 |
| methotrexate | NSC 740 |
| methotrexate derivative | NSC 174121 |
| N-(phosphonoacetyl)-L-aspartate (PALA) | NSC 224131 |
| pyrazofurin | NSC 143095 |
| trimetrexate | NSC 352122 |
DNA Antimetabolites
| 3-HP | NSC 95678 |
| 2'-deoxy-5-fluorouridine | NSC 27640 |
| 5-HP | NSC 107392 |
| alpha-TGDR | NSC 71851 |
| aphidicolin glycinate | NSC 303812 |
| ara-C | NSC 63878 |
| 5-aza-2'-deoxycytidine | NSC 127716 |
| beta-TGDR | NSC 71261 |
| cyclocytidine | NSC 145668 |
| guanazole | NSC 1895 |
| hydroxyurea | NSC 32065 |
| inosine glycodialdehyde | NSC 118994 |
| macbecin II | NSC 330500 |
| pyrazoloimidazole | NSC 51143 |
| thioguanine | NSC 752 |
| thiopurine | NSC 755 |